Trine Meldgaard Lund
Associate Professor
Translational and Clinical Pharmacology
Jagtvej 160
2100 København Ø
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Impact of the malate-aspartate shuttle in glutamate neurotransmission
Waagepetersen, Helle S., Bak, Lasse Kristoffer, Lund, Trine Meldgaard, Walls, A. B., Sonnewald, U. & Schousboe, Arne, 2009, In: Journal of Neurochemistry. s1, p. 9Research output: Contribution to journal › Conference abstract in journal › Research
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Differential localization of voltage-gated calcium channels in neurites and somata of cultured neocortical neurons.
Timmermann, D., Lund, Trine Meldgaard, Belhage, B. & Schousboe, Arne, 1999, In: Journal of Neurochemistry. 73, Suppl, p. 127 1 p.Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
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Localization and pharmacological characterization of voltage dependent calcium channels in cultured neocortical neurons
Timmermann, D. B., Lund, Trine Meldgaard, Belhage, B. & Schousboe, Arne, 2001, In: International Journal of Developmental Neuroscience. 19, 1, p. 1-10 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Modelling concentration-analgesia relationships for morphine to evaluate experimental pain models
Sverrisdóttir, E., Foster, D. J. R., Upton, R. N., Olesen, A. E., Lund, Trine Meldgaard, Gabel-Jensen, C., Drewes, A. M., Christrup, Lona Louring & Kreilgaard, M., 23 Jan 2015, In: European Journal of Pharmaceutical Sciences. 66, p. 50-58 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Pharmacokinetic Metamodel of Morphine and Morphine-6-Glucuronide in Neonates and Adults
Sverrisdóttir, E., Foster, D. J. R., Olesen, A. E., Lund, Trine Meldgaard, Drewes, A. M., Christrup, Lona Louring, Kreilgaard, M. & Upton, R. N., Jun 2016.Research output: Contribution to conference › Poster › Research
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Modelling analgesia-concentration relationships for morphine to evaluate experimental pain models
Sverrisdóttir, E., Foster, D., Upton, R., Olesen, A. E., Lund, Trine Meldgaard, Christrup, Lona Louring & Kreilgaard, M., 2013, Population Approach Group in Europe.Research output: Other contribution › Research
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Modelling analgesia-concentration relationships for morphine to evaluate experimental pain models
Sverrisdóttir, E., Foster, D., Upton, R., Olesen, A. E., Lund, Trine Meldgaard, Christrup, Lona Louring & Kreilgaard, M., Jun 2013.Research output: Contribution to conference › Poster › Research
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A review of morphine and morphine-6-glucuronide's pharmacokinetic-pharmacodynamic relationships in experimental and clinical pain
Sverrisdóttir, E., Lund, Trine Meldgaard, Olesen, A. E., Drewes, A. M., Christrup, Lona Louring & Kreilgaard, M., 7 Apr 2015, In: European Journal of Pharmaceutical Sciences. 74, p. 45–62 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Population pharmacokinetic-pharmacodynamic model of subcutaneous bupivacaine in a novel extended-release microparticle formulation
Storgaard, Ida Klitzing, Jensen, E. K., Bøgevig, S., Balchen, T., Springborg, A. H., Royal, M. A., Møller, Kirsten, Werner, M. U. & Lund, Trine Meldgaard, 2024, In: Basic & clinical pharmacology & toxicology. 134, 5, p. 676-685Research output: Contribution to journal › Journal article › Research › peer-review
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High-dose naloxone: Effects by late administration on pain and hyperalgesia following a human heat injury model. A randomized, double-blind, placebo-controlled, crossover trial with an enriched enrollment design
Springborg, A. D., Jensen, E. K., Kreilgaard, M., Petersen, M. A., Papathanasiou, T., Lund, Trine Meldgaard, Taylor, B. K. & Werner, M. U., 2020, In: PLoS ONE. 15, 11, 22 p., e0242169.Research output: Contribution to journal › Journal article › Research › peer-review
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The PHARMACOM-EPI framework for integrating pharmacometric modelling into pharmacoepidemiological research using real-world data: application to assess death associated with valproate
Soeorg, H., Sverrisdóttir, E., Andersen, Morten, Lund, Trine Meldgaard & Sessa, Maurizio, 2022, In: Clinical Pharmacology and Therapeutics. 111, 4, p. 840-856Research output: Contribution to journal › Journal article › Research › peer-review
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Pharmacom-epi: A framework for integrating pharmacometric modeling into Pharmacoepidemiological research using real-world data
Soeorg, H., Sverrisdottir, E., Andersen, Morten, Lund, Trine Meldgaard & Sessa, Maurizio, 2022, In: Pharmacoepidemiology and Drug Safety. 31, S2, p. 568-569Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
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Artificial neural network vs pharmacometric model for population prediction of plasma concentration in real-world data: a case study on valproic acid
Soeorg, H., Sverrisdóttir, E., Andersen, Morten, Lund, Trine Meldgaard & Sessa, Maurizio, 2022, In: Clinical Pharmacology and Therapeutics. 111, 6, p. 1278-1285Research output: Contribution to journal › Journal article › Research › peer-review
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Carnitine Levels in Skeletal Muscle, Blood, and Urine in Patients with Primary Carnitine Deficiency During Intermission of L-Carnitine Supplementation
Rasmussen, J., Thomsen, J. A., Olesen, J. H., Lund, Trine Meldgaard, Mohr, M., Clementsen, J., Nielsen, Olav Wendelboe & Lund, A. M., 10 Feb 2015, JIMD Reports. Zschocke, J., Baumgartner, M., Morava, E., Patterson, M., Rahman, S. & Peters, V. (eds.). Berlin: Springer, Vol. 20. p. 103-111 9 p. (JIMD Reports).Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
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KATP channel openers in the trigeminalvascular system
Ploug, K. B., Amrutkar, D. V., Baun, M., Ramachandran, R., Iversen, A., Lund, Trine Meldgaard, Gupta, S., Hay-Schmidt, A., Olesen, J. & Jansen-Olesen, I., 2012, In: Cephalagia. 32, 1Research output: Contribution to journal › Journal article › Research › peer-review
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Occurence of N-acylethanolamines and their precursors in neuronal rafts
Petersen, G., Lund, Trine Meldgaard & Hansen, Harald S., 2005, In: Chemistry and Physics of Lipids. 136, 2, p. 106-107 2 p.Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
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Quantification of the Pharmacodynamic Interaction of Morphine and Gabapentin Using a Response Surface Approach
Papathanasiou, T., Juul, R. V., Gabel-Jensen, C., Kreilgaard, M., Heegaard, Anne-Marie & Lund, Trine Meldgaard, 1 Nov 2017, In: AAPS Journal. 19, 6, p. 1804–1813 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Optimizing Dose-Finding Studies for Drug Combinations Based on Exposure-Response Models
Papathanasiou, T., Strathe, A., Overgaard, R. V., Lund, Trine Meldgaard & Hooker, A. C., 29 Jul 2019, In: The AAPS Journal. 21, 5, 95.Research output: Contribution to journal › Journal article › Research › peer-review
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Population pharmacokinetic modelling of morphine, gabapentin and their combination in the rat
Papathanasiou, T., Juul, R. V., Gabel-Jensen, C., Kreilgaard, M. & Lund, Trine Meldgaard, 2016, In: Pharmaceutical Research. 33, 11, p. 2630–2643 14 p.Research output: Contribution to journal › Journal article › Research › peer-review
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COMBINATION OF MORPHINE AND GABAPENTIN LEADS TO SYNERGISTIC EFFECTS IN A RAT MODEL OF POSTOPERATIVE PAIN
Papathanasiou, T., Juul, R. V., Heegaard, Anne-Marie, Kreilgaard, M. & Lund, Trine Meldgaard, 14 Jan 2015.Research output: Contribution to conference › Poster › Research
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Feasibility of Exposure-Response Analyses for Clinical Dose-Ranging Studies of Drug Combinations
Papathanasiou, T., Strathe, A., Hooker, A. C., Lund, Trine Meldgaard & Overgaard, R. V., May 2018, In: The AAPS Journal. 20, 13 p., 64.Research output: Contribution to journal › Journal article › Research › peer-review
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Impact of dose-escalation schemes and drug discontinuation on weight loss outcomes with liraglutide 3.0 mg: A model-based approach
Papathanasiou, T., Strathe, A., Agersø, H., Lund, Trine Meldgaard & Overgaard, R. V., 2020, In: Diabetes, Obesity and Metabolism. 22, 6, p. 969-977 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Co-administration of morphine and gabapentin leads to dose dependent synergistic effects in a rat model of postoperative pain
Papathanasiou, T., Juul, R. V., Heegaard, Anne-Marie, Kreilgaard, M. & Lund, Trine Meldgaard, 2016, In: European Journal of Pharmaceutical Sciences. 82, p. 97–105 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
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High-dose naloxone, an experimental tool uncovering latent sensitisation: pharmacokinetics in humans.
Papathanasiou, T., Springborg, A., Kongstad, Kenneth Thermann, Stærk, Dan, Møller, Kirsten, Taylor, B. K., Lund, Trine Meldgaard & Werner, M. U., 2019, In: British Journal of Anaesthesia. 123, 2, p. e204-e214Research output: Contribution to journal › Journal article › Research › peer-review
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Response surface analysis of synergistic interactions of morphine and gabapentin in a rat model of postoperative pain.
Papathanasiou, T., Juul, R. V., Heegaard, Anne-Marie, Kreilgaard, M. & Lund, Trine Meldgaard, 19 Oct 2015.Research output: Contribution to conference › Poster › Research
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Demonstrating Contribution of Components of Fixed-Dose Drug Combinations Through Longitudinal Exposure-Response Analysis
Nøhr-Nielsen, A., Lange, Theis, Forman, Julie Lyng, Papathanasiou, T., Foster, D. J. R., Upton, R. N., Bjerrum, Ole Jannik & Lund, Trine Meldgaard, 2020, In: The AAPS Journal. 22, 2, 32.Research output: Contribution to journal › Journal article › Research › peer-review
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Body of evidence and approaches applied in the clinical development programme of fixed-dose combinations in the European Union from 2010 to 2016
Nøhr-Nielsen, A., De Bruin, M. L., Thomsen, M., Pipper, C. B., Lange, Theis, Bjerrum, Ole Jannik & Lund, Trine Meldgaard, 2019, In: British Journal of Clinical Pharmacology. 85, 8, p. 1829-1840 12 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Pharmacodynamic modelling reveals synergistic interaction between docetaxel and SCO-101 in a docetaxel-resistant triple negative breast cancer cell line
Nøhr-Nielsen, A., Bagger, Sofie Morsing, Brünner, N., Stenvang, Jan & Lund, Trine Meldgaard, 2020, In: European Journal of Pharmaceutical Sciences. 148, 10 p., 105315.Research output: Contribution to journal › Journal article › Research › peer-review
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Evaluation of Multi-Frequency Bioelectrical Impedance Analysis against Dual-Energy X-ray Absorptiometry for Estimation of Low Muscle Mass in Older Hospitalized Patients
Nielsen, R. L., Andersen, A. L., Kallemose, T., Damgaard, Morten, Bornæs, O., Juul-Larsen, H. G., Strejby Christensen, L. W., Jawad, B. N., Andersen, Ove, Rasmussen, H. H., Munk, T., Lund, Trine Meldgaard & Houlind, Morten Baltzer, 2024, In: Journal of Clinical Medicine. 13, 1, 15 p., 196.Research output: Contribution to journal › Journal article › Research › peer-review
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Appetite stimulation with cannabis-based medicine and methods for assessment of glomerular filtration in older patients with medical illness: A study protocol
Nielsen, R. L., Bornæs, O., Storgaard, I. K., Kallemose, T., Jørgensen, L. M., Jawad, B. N., Altintas, I., Juul-larsen, H. G., Tavenier, J., Durhuus, J. A., Bengaard, A. K. P., Holst, J. J., Kolko, M., Sonne, D. P., Breindahl, T., Damgaard, M., Porrini, E., Hornum, M., Andersen, O., Pedersen, M. M. & 6 others, , 2023, In: Basic & Clinical Pharmacology & Toxicology. 133, 3, p. 237-253 17 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Design, synthesis and pharmacology of model compounds for indirect elucidation of the topography of AMPA receptor sites
Madsen, Ulf, Frølund, Bente, Lund, Trine Meldgaard, Ebert, B. & Krogsgaard-Larsen, Povl, 1993, In: European Journal of Medicinal Chemistry. 28, p. 791–800Research output: Contribution to journal › Journal article › Research › peer-review
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Effects of taurine depletion on cell migration and NCAM expression in cultures of dissociated mouse cerebellum and N2A cells
Maar, T. E., Lund, Trine Meldgaard, Gegelashvili, G., Hartmann-Petersen, Rasmus, Moran, M. J., Pasantes-Morales, H., Berezin, V., Bock, E. & Schousboe, Arne, 1998, In: Amino Acids. 15, 1, p. 77-88 12 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Dose Finding in the Clinical Development of 60 US Food and Drug Administration-Approved Drugs Compared With Learning vs. Confirming Recommendations
Lyauk, Y. K., Jonker, D. M. & Lund, Trine Meldgaard, 2019, In: Clinical and Translational Science. 12, 5, p. 481-489Research output: Contribution to journal › Journal article › Research › peer-review
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Integrated Item Response Theory Modeling of Multiple Patient-Reported Outcomes Assessing Lower Urinary Tract Symptoms Associated with Benign Prostatic Hyperplasia
Lyauk, Y. K., Lund, Trine Meldgaard, Hooker, A. C., Karlsson, M. O. & Jonker, D. M., 2020, In: The AAPS Journal. 22, 5, 13 p., 98.Research output: Contribution to journal › Journal article › Research › peer-review
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Item Response Theory Modeling of the International Prostate Symptom Score in Patients with Lower Urinary Tract Symptoms Associated with Benign Prostatic Hyperplasia
Lyauk, Y. K., Jonker, D. M., Lund, Trine Meldgaard, Hooker, A. C. & Karlsson, M. O., 2020, In: The AAPS Journal. 22, 5, 15 p., 115.Research output: Contribution to journal › Journal article › Research › peer-review
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Bounded Integer Modeling of Symptom Scales Specific to Lower Urinary Tract Symptoms Secondary to Benign Prostatic Hyperplasia
Lyauk, Y. K., Jonker, D. M., Hooker, A., Lund, Trine Meldgaard & Karlsson, M. O., 2021, In: The AAPS journal. 23, 2, 14 p., 33.Research output: Contribution to journal › Journal article › Research › peer-review
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AMPA receptor agonists, design, synthesis and molecular pharmacology
Lund, Trine Meldgaard, Christensen, I. T., Madsen, Ulf, Ebert, B., Brehm, L. & Krogsgaard-Larsen, Povl, 1990, In: Neurochemistry International. 16 suppl 1, 51, p. 51 1 p.Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
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Det glutamaterge system: neurokemisk patologi af Alzheimers syge og medicinalkemiske studier af glutaminsyrereceptorerne
Lund, Trine Meldgaard, 1992, 138 p. Kbh : Danmarks Farmaceutiske Højskole. Institut for Organisk Kemi.Research output: Other contribution › Research
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Availability of neurotransmitter glutamate is diminished when beta-hydroxybutyrate replaces glucose in cultured neurons
Lund, Trine Meldgaard, Risa, Ø., Sonnewald, U., Schousboe, Arne & Waagepetersen, Helle S., 2009, In: Journal of Neurochemistry. 110, 1, p. 80-91 12 p.Research output: Contribution to journal › Journal article › Research › peer-review
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The metabolic impact of β-hydroxybutyrate on neurotransmission: Reduced glycolysis mediates changes in calcium responses and KATP channel receptor sensitivity
Lund, Trine Meldgaard, Ploug, K. B., Iversen, A., Jensen, Anders A. & Jansen-Olesen, I., 2015, In: Journal of Neurochemistry. 132, 5, p. 520-531 12 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Stofskiftesygedomme - Fra gen til terapi
Lund, Trine Meldgaard, Christensen, E., Schousboe, A. & Meldgaard Lund, A., 1 Jan 2001, In: Lægemiddelforskning. p. 12-13 40 p.Research output: Contribution to journal › Journal article › Research › peer-review
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ß-Hydroxybutyrate is the preferred substrate for GABA and glutamate synthesis while glucose is indispensable during depolarization in cultured GABAergic neurons
Lund, Trine Meldgaard, Obel, L. F., Risa, Ø. & Sonnewald, U., 1 Aug 2011, In: Neurochemistry International. 59, 2, p. 309-18 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
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GABA synthesis from ß-hydroxybutyrate and glucose is differentially affected by neuronal activity in cultured GABAergic neurons
Lund, Trine Meldgaard, Risa, O., Sonnewald, U., Schousboe, Arne & Waagepetersen, Helle S., 2009, In: Journal of Neurochemistry. s2, p. 95Research output: Contribution to journal › Conference abstract in journal › Research
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ß-hydroxybutyrate and glucose metabolism is differently affected by neuronal activity
Lund, Trine Meldgaard, Clausen, M., Risa, O., Sonnewald, U., Schousboe, Arne & Waagepetersen, Helle S., 2007, In: Journal of Neurochemistry. 102, s1, p. 116Research output: Contribution to journal › Conference abstract in journal › Research
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On the neurotoxicity of glutaric, 3-hydroxyglutaric, and trans-glutaconic acids in glutaric acidemia type 1
Lund, Trine Meldgaard, Christensen, E., Kristensen, Anders Skov, Schousboe, Arne & Lund, Allan Meldgaard, 2004, In: Journal of Neuroscience Research. 77, 1, p. 143-7 5 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Aspartate-glutamate homeostasis in cerebellar neurons changes when shifting from glucose to beta-hydroxybutyrate as substrate
Lund, Trine Meldgaard, Clausen, M., Risa, Ø., Sonnewald, U., Schousboe, Arne & Waagepetersen, Helle S., 2009, In: Journal of Neurochemistry. s1, p. 291-291Research output: Contribution to journal › Conference abstract in journal › Research
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Conformational and pharmacological characterization of 4-AHCP, a bicyclic homologue of the excitatory amino acid receptor agonist AMPA
Lund, Trine Meldgaard, Madsen, Ulf, Ebert, B., Jørgensen, Flemming Steen & Krogsgaard-Larsen, Povl, 1991, In: Med. Chem. Res. 1, p. 136-141 6 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Design of excitatory amino acid receptor agonists, partial agonists and antagonists: Ibotenic acid as a key lead structure
Krogsgaard-Larsen, Povl, Ebert, B., Lund, Trine Meldgaard, Bräuner, Hans, Sloøk, F. A., Johansen, Tommy Nørskov, Brehm, L. & Madsen, Ulf, 10 Sep 1996, In: European Journal of Medicinal Chemistry. 31, 7-8, p. 515-537 23 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Excitatory amino acid receptors: multiplicity and structural requirements for activation and blockade
Krogsgaard-Larsen, Povl, Lund, Trine Meldgaard, Jørgensen, Flemming Steen & Brehn, L., 1991, Excitatory amino acids and synaptic function. Wheal, H. & Thomson, A. (eds.). London: Academic Press, p. 1-17 17 p. (Excitatory Amino Acids and Synaptic Transmission, Academic Press, London).Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
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Hydroxylated analogues of 5-aminovaleric acid as 4-aminobutyric acidB receptor antagonists: stereostructure-activity relationships
Kristiansen, Uffe, bjl587, bjl587, Herdeis, C., Lund, Trine Meldgaard, Nielsen, Birgitte, Hansen, J. J., Falch, E., Hjeds, H. & Krogsgaard-Larsen, Povl, Mar 1992, In: Journal of Neurochemistry. 58, 3, p. 1150-9 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 1303792
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Kroppens egne cannabinoider påvirker immunsystemet
Research output: Contribution to journal › Journal article › Research › peer-review
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197
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Pharmacokinetic Metamodel of Morphine and Morphine-6-Glucuronide in Neonates and Adults
Research output: Contribution to conference › Poster › Research
Published -
85
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Dose Finding in the Clinical Development of 60 US Food and Drug Administration-Approved Drugs Compared With Learning vs. Confirming Recommendations
Research output: Contribution to journal › Journal article › Research › peer-review
Published