Vladimir Shalgunov

Vladimir Shalgunov

Guest Researcher


  1. Published

    Development of Trans-Cyclooctene Modified Antibodies for Pretargeted Imaging within the Central Nervous System: [Meeting Abstract]

    van den Broek, S. L., Shalgunov, Vladimir, Sehlin, D., Syvanen, S. & Herth, Matthias Manfred, 2020, In: Journal of Nuclear Medicine. 61, Supl. 1, 3 p., 196.

    Research output: Contribution to journalConference abstract in journalResearch

  2. Published

    Transport of nanomedicines across the blood-brain barrier: Challenges and opportunities for imaging and therapy

    van den Broek, S. L., Shalgunov, Vladimir & Herth, Matthias Manfred, 2022, In: Biomaterials Advances. 141, 11 p., 213125.

    Research output: Contribution to journalReviewResearchpeer-review

  3. Published

    Development and Evaluation of Two Potential 5-HT7 Receptor PET Tracers: [18F]ENL09 and [18F]ENL10

    Tampio L'Estrade, E., Xiong, M., Shalgunov, Vladimir, Edgar, F. G., Volk, B., Baerentzen, S. L., Palner, M., Erlandsson, M., Ohlsson, T., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2019, In: ACS Chemical Neuroscience. 10, 9, p. 3961-3968 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Synthesis, Radiolabeling, and in Vitro and in Vivo Evaluation of [18F]ENL30: A Potential PET Radiotracer for the 5-HT7 Receptor

    Tampio L'Estrade, E., Edgar, F. G., Xiong, M., Shalgunov, Vladimir, Baerentzen, S. L., Erlandsson, M., Ohlsson, T. G., Palner, M., Knudsen, Gitte Moos & Herth, Matthias Manfred, 23 Apr 2019, In: ACS Omega. 4, 4, p. 7344-7353

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Fragment-based labeling using condensation reactions of six potential 5-HT7R PET tracers

    Tampio L'Estrade, E., Shalgunov, Vladimir, Lehel, S., Nymann Petersen, I., Poulie, Christian Bernard Matthijs, Edgar, F. G., Volk, B., Ohlsson, T., Erlandsson, M., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2020, In: Journal of Radioanalytical and Nuclear Chemistry. 326, p. 1749-1762 14 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Convenient Entry to 18 F-Labeled Amines through the Staudinger Reduction

    Stéen, E. J. L., Shalgunov, Vladimir, Denk, C., Mikula, H., Kjær, Andreas, Kristensen, Jesper Langgaard & Herth, Matthias Manfred, 2019, In: European Journal of Organic Chemistry. 2019, 8, p. 1722-1725

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Cover Feature: Convenient Entry to 18 F-Labeled Amines through the Staudinger Reduction (Eur. J. Org. Chem. 8/2019)

    Stéen, E. J. L., Shalgunov, Vladimir, Denk, C., Mikula, H., Kjær, Andreas, Kristensen, Jesper Langgaard & Herth, Matthias Manfred, 28 Feb 2019, In: European Journal of Organic Chemistry. 2019, 8, p. 1686-1686

    Research output: Contribution to journalJournal articleCommunication

  8. Published

    Improved radiosynthesis and preliminary in vivo evaluation of the 11 C-labeled tetrazine [ 11 C]AE-1 for pretargeted PET imaging

    Stéen, E. J. L., Jørgensen, Jesper Tranekjær, Petersen, I. N., Nørregaard, K., Lehel, S., Shalgunov, Vladimir, Birke, A., Edem, P. E., L'Estrade, E. T., Hansen, H. D., Villadsen, J., Erlandsson, M., Ohlsson, T., Yazdani, A., Valliant, J. F., Kristensen, Jesper Langgaard, Barz, M., Knudsen, Gitte Moos, Kjær, Andreas & Herth, Matthias Manfred, 1 Jan 2019, In: Bioorganic and Medicinal Chemistry Letters. 29, 8, p. 986-990

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Trans-Cyclooctene-Functionalized PeptoBrushes with Improved Reaction Kinetics of the Tetrazine Ligation for Pretargeted Nuclear Imaging

    Stéen, E. J. L., Jørgensen, Jesper Tranekjær, Johann, K., Norregaard, K., Sohr, B., Svatunek, D., Birke, A., Shalgunov, Vladimir, Edem, P. E., Rossin, R., Seidl, C., Schmid, F., Robillard, M. S., Kristensen, Jesper Langgaard, Mikula, H., Barz, M., Kjær, Andreas & Herth, Matthias Manfred, 2020, In: ACS Nano. 14, 1, p. 568-584

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Pretargeting in nuclear imaging and radionuclide therapy: Improving efficacy of theranostics and nanomedicines

    Stéen, E. J. L., Edem, P. E., Nørregaard, K., Jørgensen, Jesper Tranekjær, Shalgunov, Vladimir, Kjær, Andreas & Herth, Matthias Manfred, Oct 2018, In: Biomaterials. 179, p. 209-245 37 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    Lipophilicity and Click Reactivity Determine the Performance of Bioorthogonal Tetrazine Tools in Pretargeted In Vivo Chemistry

    Steen, E. J. L., Jørgensen, Jesper Tranekjær, Denk, C., Battisti, Umberto Maria, Norregaard, K., Edem, P. E., Bratteby, K., Shalgunov, Vladimir, Wilkovitsch, M., Svatunek, D., Poulie, Christian Bernard Matthijs, Hvass, Lars, Simon, M., Wanek, T., Rossin, R., Robillard, M., Kristensen, Jesper Langgaard, Mikula, H., Kjær, Andreas & Herth, Matthias Manfred, 2021, In: ACS Pharmacology & Translational Science. 4, 2, p. 824-833 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    Development of 11C-labeled CRANAD-102 for positron emission tomography imaging of soluble Aβ-species

    Staudt, Markus, Shalgunov, Vladimir, Nedergaard, Maiken & Herth, Matthias Manfred, 2023, In: Journal of Labelled Compounds and Radiopharmaceuticals. 66, 12, p. 393-399

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Published

    A SPECT-based method for dynamic imaging of the glymphatic system in rats

    Sigurdsson, B., Hauglund, Natalie Linea, Lilius, T. O., Mogensen, F. L. H., Mortensen, K. N., Beschorner, Natalie, Klinger, L., Bærentzen, S. L., Rosenholm, Marko, Shalgunov, Vladimir, Herth, Matthias Manfred, Mori, Yuki & Nedergaard, Maiken, 2023, In: Journal of Cerebral Blood Flow and Metabolism. 43, 7, 13 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  14. Published

    Blocking of efflux transporters in rats improves translational validation of brain radioligands

    Shalgunov, Vladimir, Xiong, M., L’Estrade, E. T., Raval, N. R., Andersen, Ida Vang, Edgar, F. G., Speth, N. R., Baerentzen, S. L., Hansen, H. D., Donovan, L. L., Nasser, A., Peitersen, S. T., Kjær, Andreas, Knudsen, Gitte Moos, Syvänen, S., Palner, M. & Herth, Matthias Manfred, 2020, In: EJNMMI Research. 10, 1, 11 p., 124.

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    Evaluation of F-537-Tetrazine in a model for brain pretargeting imaging. Comparison to N-(3-[18F] fluoro-5-(1,2,4,5-tetrazin-3-yl)benzyl)propan-1-amine

    Shalgunov, Vladimir, van den Broek, S. L., Andersen, Ida Vang, Raval, N. R., Schäfer, G., Barz, M., Herth, Matthias Manfred & Battisti, Umberto Maria, 2024, In: Nuclear Medicine and Biology. 128-129, 12 p., 108877.

    Research output: Contribution to journalJournal articleResearchpeer-review

  16. Published

    Convenient access to F-18-labeled amines through the Staudinger reduction

    Shalgunov, Vladimir, Steen, J., Denk, C., Mikula, H., Kjær, Andreas, Kristensen, Jesper Langgaard & Herth, Matthias Manfred, May 2019, In: Journal of Labelled Compounds and Radiopharmaceuticals. 62, Supl. 1/SI, p. S205-S206 P-050.

    Research output: Contribution to journalConference abstract in journalResearch

  17. Hunting for the high-affinity state of G-protein-coupled receptors with agonist tracers: Theoretical and practical considerations for positron emission tomography imaging

    Shalgunov, Vladimir, van Waarde, A., Booij, J., Michel, M. C., Dierckx, R. A. J. O. & Elsinga, P. H., May 2019, In: Medicinal Research Reviews. 39, 3, p. 1014-1052

    Research output: Contribution to journalReviewResearchpeer-review

  18. Published

    SPECT imaging of the glymphatic pathway with In-111-labeled ovalbumin in the rat brain

    Shalgunov, Vladimir, Lilius, T., Sigurosson, B., Baerentzen, S. L., Hauglund, Natalie Linea, Herth, Matthias Manfred, Palner, M. & Nedergaard, Maiken, 2019, In: Journal of Labelled Compounds and Radiopharmaceuticals. 62, Supplement 1, p. S404-S405 2 p.

    Research output: Contribution to journalConference abstract in journalResearchpeer-review

  19. Published

    Radiolabeling of a polypeptide polymer for intratumoral delivery of alpha-particle emitter, 225Ac, and beta-particle emitter, 177Lu

    Shalgunov, Vladimir, Engudar, G., Bohrmann, L., Wharton, L., Maskell, K., Johann, K., Barz, M., Schaffer, P., Herth, Matthias Manfred & Radchenko, V., 2022, In: Nuclear Medicine and Biology. 104-105, p. 11-21

    Research output: Contribution to journalJournal articleResearchpeer-review

  20. Published

    Preliminary Evaluation of (S)-7-[F-18]Fluorotryptophan as a Tracer for the Imaging of Serotonin Synthesis in Pig Brain

    Shalgunov, Vladimir, Raval, N. R., Donovan, L. L., Nasser, A., Zlatopolskiy, B. D., Neumaier, B., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2020, In: European Journal of Nuclear Medicine and Molecular Imaging. 47, SUPPL 1, p. S639-S639 EP-267 .

    Research output: Contribution to journalConference abstract in journalResearchpeer-review

  21. Published

    Evaluation of the α-synuclein PET radiotracer (d3)-[11C]MODAG-001 in pigs

    Raval, N. R., Madsen, C. A., Shalgunov, Vladimir, Nasser, A., Battisti, Umberto Maria, Beaman, Emily Eufaula, Juhl, M., Jørgensen, Louise Møller, Herth, Matthias Manfred, Hansen, H. D., Plavén-Sigray, P. & Knudsen, Gitte Moos, 2022, In: Nuclear Medicine and Biology. 114-115, p. 42-48

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. Published

    Development of the First Tritiated Tetrazine: Facilitating Tritiation of Proteins

    Radjani Bidesi, N. S., Battisti, Umberto Maria, Lopes van de Broek, S., Shalgunov, Vladimir, Dall, A., Bøggild Kristensen, J., Sehlin, D., Syvänen, S., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2022, In: ChemBioChem. 23, 23, 7 p., e202200539.

    Research output: Contribution to journalJournal articleResearchpeer-review

  23. Published

    Bioorthogonal Click of Colloidal Gold Nanoparticles to Antibodies In vivo

    Poulie, Christian Bernard Matthijs, Sporer, E., Hvass, Lars, Jørgensen, Jesper Tranekjær, Kempen, Paul Joseph, Lopes van den Broek, S. I., Shalgunov, Vladimir, Kjær, Andreas, Jensen, A. I. & Herth, Matthias Manfred, 2022, In: Chemistry - A European Journal. 28, 61, 10 p., e202201847.

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    Next generation fibroblast activation protein (FAP) targeting PET tracers : The tetrazine ligation allows an easy and convenient way to 18F-labeled (4-quinolinoyl)glycyl-2-cyanopyrrolidines

    Poulie, Christian Bernard Matthijs, Shalgunov, Vladimir, Elvas, F., Van Rymenant, Y., Moon, E. S., Battisti, Umberto Maria, De Loose, J., De Meester, I., Rösch, F., Van Der Veken, P. & Herth, Matthias Manfred, 2023, In: European Journal of Medicinal Chemistry. 262, 10 p., 115862.

    Research output: Contribution to journalJournal articleResearchpeer-review

  25. Published

    Evaluation of [Cu-64]Cu-NOTA-PEG7-H-Tz for Pretargeted Imaging in LS174T Xenografts-Comparison to [111In-111]In-DOTA-PEG11-BisPy-Tz

    Poulie, Christian Bernard Matthijs, Jørgensen, Jesper Tranekjær, Shalgunov, Vladimir, Kougioumtzoglou, G., Jeppesen, T. E., Kjær, Andreas & Herth, Matthias Manfred, 2021, In: Molecules. 26, 3, 9 p., 544.

    Research output: Contribution to journalJournal articleResearchpeer-review

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ID: 185059116