Vladimir Shalgunov
Guest Researcher
Medicinal Chemistry
Jagtvej 162
2100 København Ø
- 2018
- Published
Pretargeting in nuclear imaging and radionuclide therapy: Improving efficacy of theranostics and nanomedicines
Stéen, E. J. L., Edem, P. E., Nørregaard, K., Jørgensen, Jesper Tranekjær, Shalgunov, Vladimir, Kjær, Andreas & Herth, Matthias Manfred, Oct 2018, In: Biomaterials. 179, p. 209-245 37 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2019
- Published
Convenient Entry to 18 F-Labeled Amines through the Staudinger Reduction
Stéen, E. J. L., Shalgunov, Vladimir, Denk, C., Mikula, H., Kjær, Andreas, Kristensen, Jesper Langgaard & Herth, Matthias Manfred, 2019, In: European Journal of Organic Chemistry. 2019, 8, p. 1722-1725Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Development and Evaluation of Two Potential 5-HT7 Receptor PET Tracers: [18F]ENL09 and [18F]ENL10
Tampio L'Estrade, E., Xiong, M., Shalgunov, Vladimir, Edgar, F. G., Volk, B., Baerentzen, S. L., Palner, M., Erlandsson, M., Ohlsson, T., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2019, In: ACS Chemical Neuroscience. 10, 9, p. 3961-3968 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
High-throughput rat brain PET imaging and automatic spatial normalization of the dopamine D2/3 receptor ligand [F-18]fallypride
Lange, D., Tejada, I. M., Xiong, M., Hillebrand, B., Noergaard, M., Baerentzen, S., Shalgunov, Vladimir, Herth, Matthias Manfred, Svarer, C. & Palner, M., 2019, In: Journal of Cerebral Blood Flow and Metabolism. 39, p. 588-589 2 p.Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
- Published
SPECT imaging of the glymphatic pathway with In-111-labeled ovalbumin in the rat brain
Shalgunov, Vladimir, Lilius, T., Sigurosson, B., Baerentzen, S. L., Hauglund, Natalie Linea, Herth, Matthias Manfred, Palner, M. & Nedergaard, Maiken, 2019, In: Journal of Labelled Compounds and Radiopharmaceuticals. 62, Supplement 1, p. S404-S405 2 p.Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
- Published
The Chemogenetic Receptor Ligand Clozapine N-Oxide Induces in vivo Neuroreceptor Occupancy and Reduces Striatal Glutamate Levels
Bærentzen, S., Casado-Sainz, A., Lange, D., Shalgunov, Vladimir, Tejada, I. M., Xiong, M., L'Estrade, E. T., Edgar, F. G., Lee, H., Herth, Matthias Manfred & Palner, M., 2019, In: Frontiers in Neuroscience. 13, 7 p., 187.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The polypharmacological profile of psilocybin and potential behavioural effects of very low doses
Kiilerich, K., Speth, N., Lorenz, J., Casado-Sainz, A., Shalgunov, Vladimir, Lange, D., Xiong, M., Herth, Matthias Manfred, Overgaard, A., Hansen, H. D. & Palner, M., 2019, In: European Neuropsychopharmacology. 29, Supplement 6, p. S175-S176 2 p.Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
- Published
Improved radiosynthesis and preliminary in vivo evaluation of the 11 C-labeled tetrazine [ 11 C]AE-1 for pretargeted PET imaging
Stéen, E. J. L., Jørgensen, Jesper Tranekjær, Petersen, I. N., Nørregaard, K., Lehel, S., Shalgunov, Vladimir, Birke, A., Edem, P. E., L'Estrade, E. T., Hansen, H. D., Villadsen, J., Erlandsson, M., Ohlsson, T., Yazdani, A., Valliant, J. F., Kristensen, Jesper Langgaard, Barz, M., Knudsen, Gitte Moos, Kjær, Andreas & Herth, Matthias Manfred, 1 Jan 2019, In: Bioorganic and Medicinal Chemistry Letters. 29, 8, p. 986-990Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Cover Feature: Convenient Entry to 18 F-Labeled Amines through the Staudinger Reduction (Eur. J. Org. Chem. 8/2019)
Stéen, E. J. L., Shalgunov, Vladimir, Denk, C., Mikula, H., Kjær, Andreas, Kristensen, Jesper Langgaard & Herth, Matthias Manfred, 28 Feb 2019, In: European Journal of Organic Chemistry. 2019, 8, p. 1686-1686Research output: Contribution to journal › Journal article › Communication
- Published
Synthesis, Radiolabeling, and in Vitro and in Vivo Evaluation of [18F]ENL30: A Potential PET Radiotracer for the 5-HT7 Receptor
Tampio L'Estrade, E., Edgar, F. G., Xiong, M., Shalgunov, Vladimir, Baerentzen, S. L., Erlandsson, M., Ohlsson, T. G., Palner, M., Knudsen, Gitte Moos & Herth, Matthias Manfred, 23 Apr 2019, In: ACS Omega. 4, 4, p. 7344-7353Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Convenient access to F-18-labeled amines through the Staudinger reduction
Shalgunov, Vladimir, Steen, J., Denk, C., Mikula, H., Kjær, Andreas, Kristensen, Jesper Langgaard & Herth, Matthias Manfred, May 2019, In: Journal of Labelled Compounds and Radiopharmaceuticals. 62, Supl. 1/SI, p. S205-S206 P-050.Research output: Contribution to journal › Conference abstract in journal › Research
- Published
F-18-Radiolabeling and in vivo evaluation of two diverse glycomimetics using PET
Bratteby, K., Torkelsson, E., L'Estrade, E. T., Peterson, K., Shalgunov, Vladimir, Xiong, M., Leffer, H., Zetterberg, F., Ohlsson, T., Gillings, N., Nilsson, U., Herth, Matthias Manfred & Erlandsson, M., May 2019, p. S533-S534.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
Hunting for the high-affinity state of G-protein-coupled receptors with agonist tracers: Theoretical and practical considerations for positron emission tomography imaging
Shalgunov, Vladimir, van Waarde, A., Booij, J., Michel, M. C., Dierckx, R. A. J. O. & Elsinga, P. H., May 2019, In: Medicinal Research Reviews. 39, 3, p. 1014-1052Research output: Contribution to journal › Review › Research › peer-review
- Published
PET radiotracer translation from rats to higher species, using an increased-throughput in vivo evaluation strategy
L'Estrade, E. T., Xiong, M., Petersen, I., Shalgunov, Vladimir, Edgar, F. G., Hansen, H., Erlandsson, M., Ohlsson, T., Knudsen, Gitte Moos, Palner, M. & Herth, Matthias Manfred, May 2019, p. S389-S390.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
- 2020
- Published
Blocking of efflux transporters in rats improves translational validation of brain radioligands
Shalgunov, Vladimir, Xiong, M., L’Estrade, E. T., Raval, N. R., Andersen, Ida Vang, Edgar, F. G., Speth, N. R., Baerentzen, S. L., Hansen, H. D., Donovan, L. L., Nasser, A., Peitersen, S. T., Kjær, Andreas, Knudsen, Gitte Moos, Syvänen, S., Palner, M. & Herth, Matthias Manfred, 2020, In: EJNMMI Research. 10, 1, 11 p., 124.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Development of Trans-Cyclooctene Modified Antibodies for Pretargeted Imaging within the Central Nervous System: [Meeting Abstract]
van den Broek, S. L., Shalgunov, Vladimir, Sehlin, D., Syvanen, S. & Herth, Matthias Manfred, 2020, In: Journal of Nuclear Medicine. 61, Supl. 1, 3 p., 196.Research output: Contribution to journal › Conference abstract in journal › Research
- Published
Fragment-based labeling using condensation reactions of six potential 5-HT7R PET tracers
Tampio L'Estrade, E., Shalgunov, Vladimir, Lehel, S., Nymann Petersen, I., Poulie, Christian Bernard Matthijs, Edgar, F. G., Volk, B., Ohlsson, T., Erlandsson, M., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2020, In: Journal of Radioanalytical and Nuclear Chemistry. 326, p. 1749-1762 14 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
In Vivo Veritas - 18F-radiolabeled glycomimetics allow insights into the pharmacological fate of galectin-3 inhibitors
Bratteby, K., Torkelsson, E., Tampio L'Estrade, E., Peterson, K., Shalgunov, Vladimir, Xiong, M., Leffler, H., Zetterberg, F., Olsson, T. G., Gillings, N., Nilsson, U. J., Herth, Matthias Manfred & Erlandsson, M., 2020, In: Journal of Medicinal Chemistry. 63, 2, p. 747-755Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Preliminary Evaluation of (S)-7-[F-18]Fluorotryptophan as a Tracer for the Imaging of Serotonin Synthesis in Pig Brain
Shalgunov, Vladimir, Raval, N. R., Donovan, L. L., Nasser, A., Zlatopolskiy, B. D., Neumaier, B., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2020, In: European Journal of Nuclear Medicine and Molecular Imaging. 47, SUPPL 1, p. S639-S639 EP-267 .Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
- Published
Preliminary Evaluation of (S)-7-[F-18]Fluorotryptophan as a Tracer for the Imaging of Tryptophan Metabolism Alterations in Tumor Xenografts
Hvass, L., Shalgunov, Vladimir, Jorgensen, J. T., Zlatopolskiy, B. D., Neumaier, B., Kjær, Andreas & Herth, Matthias Manfred, 2020, In: European Journal of Nuclear Medicine and Molecular Imaging. 47, SUPPL 1, p. S646-S647 Meeting Abstract: EP-282 .Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
- Published
Radiosynthesis and preclinical evaluation of [11 C]Cimbi-701 - Towards the imaging of cerebral 5-HT7 receptors
L 'Estrade, E. T., Shalgunov, Vladimir, Edgar, F. G., Strebl-Bantillo, M. G., Xiong, M., Crestey, F., Neelamegam, R., Dyssegaard, A., Lehel, S., Erlandsson, M., Ohlsson, T., Hooker, J. M., Knudsen, Gitte Moos, Herth, Matthias Manfred & Hansen, H. D., 2020, In: Journal of Labelled Compounds and Radiopharmaceuticals. 63, p. 46-55Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Trans-Cyclooctene-Functionalized PeptoBrushes with Improved Reaction Kinetics of the Tetrazine Ligation for Pretargeted Nuclear Imaging
Stéen, E. J. L., Jørgensen, Jesper Tranekjær, Johann, K., Norregaard, K., Sohr, B., Svatunek, D., Birke, A., Shalgunov, Vladimir, Edem, P. E., Rossin, R., Seidl, C., Schmid, F., Robillard, M. S., Kristensen, Jesper Langgaard, Mikula, H., Barz, M., Kjær, Andreas & Herth, Matthias Manfred, 2020, In: ACS Nano. 14, 1, p. 568-584Research output: Contribution to journal › Journal article › Research › peer-review
- 2021
- Published
Aliphatic 18F-Radiofluorination: Recent Advances in the Labeling of Base-Sensitive Substrates**
Bratteby, K., Shalgunov, Vladimir & Herth, Matthias Manfred, 2021, In: ChemMedChem. 16, 17, p. 2612-2622Research output: Contribution to journal › Review › Research › peer-review
- Published
Development of the First Aliphatic 18F-Labeled Tetrazine Suitable for Pretargeted PET Imaging-Expanding the Bioorthogonal Tool Box
Battisti, Umberto Maria, Bratteby, K., Jørgensen, Jesper Tranekjær, Hvass, Lars, Shalgunov, Vladimir, Mikula, H., Kjær, Andreas & Herth, Matthias Manfred, 2021, In: Journal of Medicinal Chemistry. 64, 20, p. 15297–15312Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Direct Cu-mediated aromatic18F-labeling of highly reactive tetrazines for pretargeted bioorthogonal PET imaging
García-Vázquez, R., Battisti, Umberto Maria, Jørgensen, Jesper Tranekjær, Shalgunov, Vladimir, Hvass, Lars, Stares, D. L., Petersen, I. N., Crestey, F., Löffler, A., Svatunek, D., Kristensen, Jesper Langgaard, Mikula, H., Kjær, Andreas & Herth, Matthias Manfred, 2021, In: Chemical Science. 12, 35, p. 11668-11675Research output: Contribution to journal › Journal article › Research › peer-review
ID: 185059116
Most downloads
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580
downloads
SPECT imaging of the glymphatic pathway with In-111-labeled ovalbumin in the rat brain
Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
Published -
551
downloads
Convenient access to F-18-labeled amines through the Staudinger reduction
Research output: Contribution to journal › Conference abstract in journal › Research
Published -
369
downloads
Pretargeting in nuclear imaging and radionuclide therapy: Improving efficacy of theranostics and nanomedicines
Research output: Contribution to journal › Journal article › Research › peer-review
Published