4-Acylamino-and 4-ureidobenzamides as melanin-concentrating hormone (MCH) receptor 1 antagonists
Research output: Contribution to journal › Journal article › Research › peer-review
Synthesis, in vitro biological evaluation and structure-activity relationships of 4-acylamino-and 4-ureidobenzamides as novel hMCH1R-antagonists are disclosed. The nature of the amine side chains could be varied considerably in contrast to the central benzamide scaffold and aromatic substituents.
| Original language | English |
|---|---|
| Journal | Bioorganic & Medicinal Chemistry Letters |
| Volume | 14 |
| Issue number | 20 |
| Pages (from-to) | 5075-5080 |
| Number of pages | 6 |
| ISSN | 0960-894X |
| DOIs | |
| Publication status | Published - 18 Oct 2004 |
- Animals, Benzamides, CHO Cells, Cricetinae, Cricetulus, Humans, Hypothalamic Hormones, Ligands, Melanins, Pituitary Hormones, Radioligand Assay, Receptors, Pituitary Hormone, Structure-Activity Relationship, Urea
Research areas
ID: 189159527