Expedient protocol for solid-phase synthesis of secondary and tertiary amines

Research output: Contribution to journal › Journal article › Research › peer-review

Standard

Expedient protocol for solid-phase synthesis of secondary and tertiary amines. / Olsen, Christian A; Witt, Matthias; Jaroszewski, Jerzy W; Franzyk, Henrik.

In: Organic Letters, Vol. 6, No. 12, 2004, p. 1935-8.

Research output: Contribution to journal › Journal article › Research › peer-review

Harvard

Olsen, CA, Witt, M, Jaroszewski, JW & Franzyk, H 2004, 'Expedient protocol for solid-phase synthesis of secondary and tertiary amines', Organic Letters, vol. 6, no. 12, pp. 1935-8. https://doi.org/10.1021/ol049575h

APA

Olsen, C. A., Witt, M., Jaroszewski, J. W., & Franzyk, H. (2004). Expedient protocol for solid-phase synthesis of secondary and tertiary amines. Organic Letters, 6(12), 1935-8. https://doi.org/10.1021/ol049575h

Vancouver

Olsen CA, Witt M, Jaroszewski JW, Franzyk H. Expedient protocol for solid-phase synthesis of secondary and tertiary amines. Organic Letters. 2004;6(12):1935-8. https://doi.org/10.1021/ol049575h

Author

Olsen, Christian A ; Witt, Matthias ; Jaroszewski, Jerzy W ; Franzyk, Henrik. / Expedient protocol for solid-phase synthesis of secondary and tertiary amines. In: Organic Letters. 2004 ; Vol. 6, No. 12. pp. 1935-8.

Bibtex

@article{63212ce7935541c8b2edfcee8a806307,
title = "Expedient protocol for solid-phase synthesis of secondary and tertiary amines",
abstract = "[reaction: see text] An expedient solid-phase synthetic approach to secondary and tertiary amines was developed. The protocol employs conversion of resin-bound amino alcohols to the corresponding iodides, followed by iodide displacement with primary or secondary amines or with unprotected amino alcohols. This two-step procedure, affording products in good to excellent yields, is suitable for solid-phase synthesis of polyamines.",
author = "Olsen, {Christian A} and Matthias Witt and Jaroszewski, {Jerzy W} and Henrik Franzyk",
year = "2004",
doi = "10.1021/ol049575h",
language = "English",
volume = "6",
pages = "1935--8",
journal = "Organic Letters",
issn = "1523-7060",
publisher = "American Chemical Society",
number = "12",

}

RIS

TY - JOUR

T1 - Expedient protocol for solid-phase synthesis of secondary and tertiary amines

AU - Olsen, Christian A

AU - Witt, Matthias

AU - Jaroszewski, Jerzy W

AU - Franzyk, Henrik

PY - 2004

Y1 - 2004

N2 - [reaction: see text] An expedient solid-phase synthetic approach to secondary and tertiary amines was developed. The protocol employs conversion of resin-bound amino alcohols to the corresponding iodides, followed by iodide displacement with primary or secondary amines or with unprotected amino alcohols. This two-step procedure, affording products in good to excellent yields, is suitable for solid-phase synthesis of polyamines.

AB - [reaction: see text] An expedient solid-phase synthetic approach to secondary and tertiary amines was developed. The protocol employs conversion of resin-bound amino alcohols to the corresponding iodides, followed by iodide displacement with primary or secondary amines or with unprotected amino alcohols. This two-step procedure, affording products in good to excellent yields, is suitable for solid-phase synthesis of polyamines.

U2 - 10.1021/ol049575h

DO - 10.1021/ol049575h

M3 - Journal article

C2 - 15176787

VL - 6

SP - 1935

EP - 1938

JO - Organic Letters

JF - Organic Letters

SN - 1523-7060

IS - 12

ER -

ID: 42380794