Solid-phase polyamine synthesis using piperazine and piperidine building blocks

Research output: Contribution to journal › Journal article › Research › peer-review

Standard

Solid-phase polyamine synthesis using piperazine and piperidine building blocks. / Olsen, Christian A; Witt, Matthias; Jaroszewski, Jerzy W; Franzyk, Henrik.

In: Organic Letters, Vol. 5, No. 22, 2003, p. 4183-5.

Research output: Contribution to journal › Journal article › Research › peer-review

Harvard

Olsen, CA, Witt, M, Jaroszewski, JW & Franzyk, H 2003, 'Solid-phase polyamine synthesis using piperazine and piperidine building blocks', Organic Letters, vol. 5, no. 22, pp. 4183-5. https://doi.org/10.1021/ol035610t

APA

Olsen, C. A., Witt, M., Jaroszewski, J. W., & Franzyk, H. (2003). Solid-phase polyamine synthesis using piperazine and piperidine building blocks. Organic Letters, 5(22), 4183-5. https://doi.org/10.1021/ol035610t

Vancouver

Olsen CA, Witt M, Jaroszewski JW, Franzyk H. Solid-phase polyamine synthesis using piperazine and piperidine building blocks. Organic Letters. 2003;5(22):4183-5. https://doi.org/10.1021/ol035610t

Author

Olsen, Christian A ; Witt, Matthias ; Jaroszewski, Jerzy W ; Franzyk, Henrik. / Solid-phase polyamine synthesis using piperazine and piperidine building blocks. In: Organic Letters. 2003 ; Vol. 5, No. 22. pp. 4183-5.

Bibtex

@article{d9f6fea747d44821af3fddba4d4967e7,
title = "Solid-phase polyamine synthesis using piperazine and piperidine building blocks",
abstract = "[reaction: see text]. Polyamines containing piperidine and piperazine moieties have been synthesized on solid support using SN2 alkylation of resin-bound secondary amines with 2-nitrobenzenesulfonates (nosylates). The effect of solvent on this alkylation was investigated. The methodology was employed for the total synthesis of novel analogues of wasp polyamine toxins (philanthotoxins).",
author = "Olsen, {Christian A} and Matthias Witt and Jaroszewski, {Jerzy W} and Henrik Franzyk",
year = "2003",
doi = "10.1021/ol035610t",
language = "English",
volume = "5",
pages = "4183--5",
journal = "Organic Letters",
issn = "1523-7060",
publisher = "American Chemical Society",
number = "22",

}

RIS

TY - JOUR

T1 - Solid-phase polyamine synthesis using piperazine and piperidine building blocks

AU - Olsen, Christian A

AU - Witt, Matthias

AU - Jaroszewski, Jerzy W

AU - Franzyk, Henrik

PY - 2003

Y1 - 2003

N2 - [reaction: see text]. Polyamines containing piperidine and piperazine moieties have been synthesized on solid support using SN2 alkylation of resin-bound secondary amines with 2-nitrobenzenesulfonates (nosylates). The effect of solvent on this alkylation was investigated. The methodology was employed for the total synthesis of novel analogues of wasp polyamine toxins (philanthotoxins).

AB - [reaction: see text]. Polyamines containing piperidine and piperazine moieties have been synthesized on solid support using SN2 alkylation of resin-bound secondary amines with 2-nitrobenzenesulfonates (nosylates). The effect of solvent on this alkylation was investigated. The methodology was employed for the total synthesis of novel analogues of wasp polyamine toxins (philanthotoxins).

U2 - 10.1021/ol035610t

DO - 10.1021/ol035610t

M3 - Journal article

C2 - 14572280

VL - 5

SP - 4183

EP - 4185

JO - Organic Letters

JF - Organic Letters

SN - 1523-7060

IS - 22

ER -

ID: 42385442