Synthesis and Selective Functionalization of [1,2,4]Triazolo[4,3-a]pyrazines

Research output: Contribution to journalLetterResearchpeer-review

  • Charles Sylvain Demmer
  • Morten Jorgensen
  • Jan Kehler
  • Bunch, Lennart
  • Lars K. Rasmussen
A new tactic for the synthesis and selective functionalization of [1,2,4]triazolo[4,3-a]pyrazines has been developed using an oxidative cyclization as key step. Furthermore, novel strategies for introducing diverse substituents in all positions of the heterocycle were identified.
Original languageEnglish
JournalSYNLETT: Accounts and Rapid Communications in Chemical Synthesis
Volume26
Issue number4
Pages (from-to)519-524
Number of pages6
ISSN0936-5214
DOIs
Publication statusPublished - 2015

    Research areas

  • heterocyclic chemistry, cyclization, lithiation, cross-coupling, PhI(OAc)(2)

ID: 134791921