Uffe Kristiansen
Associate Professor
Molecular and Cellular Pharmacology
Jagtvej 160
2100 København Ø
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The sodium channel activator Lu AE98134 normalizes the altered firing properties of fast spiking interneurons in Dlx5/6+/- mice
von Schoubye, N. L., Frederiksen, K., Kristiansen, Uffe, Petersen, A. V., Dalby, N. O., Grunnet, M., Jensen, H. S., Jespersen, Thomas, Sohal, V. S. & Perrier, Jean-Francois Marie, 2018, In: Neuroscience Letters. 662, p. 29-35 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Direct Optical Detection of Singlet Oxygen from a Single Cell
Zebger, I., Snyder, J. W., Andersen, L. K., Poulsen, L., Gao, Z., Lambert, J. D. C., Kristiansen, Uffe & Ogilby, P. R., Apr 2004, In: Photochemistry and Photobiology. 79, 4, p. 319-322 4 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Differences in kinetics of structurally related competitive GABAA receptor antagonists
Vestergaard, H. T., Cannillo, C., Frølund, Bente & Kristiansen, Uffe, 2007, In: Neuropharmacology. 52, 3, p. 873-882Research output: Contribution to journal › Journal article › Research › peer-review
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Long-term immune cell profiling in stroke patients with or without infections
Sørensen, N. V., Hasseldam, Henrik, Johansen, F. F., Kristiansen, Uffe, Overgaard, K., Iversen, Helle Klingenberg & Rasmussen, Rune Skovgaard, 2024, In: International Journal of Neuroscience. 134, 2, p. 197-205Research output: Contribution to journal › Journal article › Research › peer-review
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Anticonvulsive evaluation of THIP in the murine pentylenetetrazole kindling model: lack of anticonvulsive effect of THIP despite functional δ-subunit-containing GABAA receptors in dentate gyrus granule cells
Simonsen, C., Boddum, K., von Schoubye, N. L., Kloppenburg, A., Sønderskov, K., Hansen, S. L. & Kristiansen, Uffe, Aug 2017, In: Pharmacology Research & Perspectives. 5, 4, 15 p., e00322.Research output: Contribution to journal › Journal article › Research › peer-review
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Effect of Rhoicissus digitata extracts on acetylcholine-mediated contraction in rat uterus
Schou, J., Kristiansen, Uffe, Stafford, G. I., van Heerden, F. & Jäger, A., Aug 2010, In: Planta Medica. 76, 12, p. 1217Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
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Acute but not delayed amphetamine treatment improves behavioral outcome in a rat embolic stroke model
Rasmussen, Rune Skovgaard, Overgaard, K., Kristiansen, Uffe & Johansen, F. F., Sep 2011, In: Neurological Research. 33, 7, p. 774-782 14 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Synthesis and biological evaluation of 4-(aminomethyl)-1-hydroxypyrazole analogues of muscimol as ¿-aminobutyric acidA receptor agonists
Petersen, J. G., Bergmann, R., Møller, H. A., Jørgensen, Charlotte Grube, Nielsen, Birgitte, Kehler, J., Frydenvang, Karla Andrea, Kristensen, Jesper Langgaard, Balle, T., Jensen, Anders A., Kristiansen, Uffe & Frølund, Bente, 2013, In: Journal of Medicinal Chemistry. 56, 3, p. 993-1006Research output: Contribution to journal › Journal article › Research › peer-review
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Uterine contraction induced by Tanzanian plants used to induce abortion
Nikolajsen, T., Nielsen, F., Rasch, V., Sørensen, P. H., Ismail, F., Kristiansen, Uffe & Jäger, A. K., 1 Sep 2011, In: Journal of Ethnopharmacology. 137, 1, p. 921-925Research output: Contribution to journal › Journal article › Research › peer-review
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Activation on single heteromeric GABAA receptor Ion channels by full and partial agonists
Mortensen, M., Kristiansen, Uffe, Ebert, B., Frølund, Bente, Krogsgaard-Larsen, Povl & Smart, T., 2004, In: Journal of Physiology. p. 393–417Research output: Contribution to journal › Journal article › Research › peer-review
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Activation of single heteromeric GABAA receptor ion channels by full and partial agonists
Mortensen, M., Kristiansen, Uffe, Ebert, B., Frølund, Bente, Krogsgaard-Larsen, Povl & Smart, T. G., 1 Jun 2004, In: Journal of Physiology. 557, 2, p. 389-413 25 p.Research output: Contribution to journal › Journal article › Research › peer-review
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5-Substituted imidazole-4-acetic acid analogues: Synthesis, modeling, and pharmacological characterization of a series of novel γ-aminobutyric acidC receptor agonists
Madsen, C., Jensen, Anders A., Liljefors, T., Kristiansen, Uffe, Nielsen, Birgitte, Hansen, C. P., Larsen, M., Ebert, B., Bang-Andersen, B., Krogsgaard-Larsen, Povl & Frølund, Bente, 2007, In: Journal of Medicinal Chemistry. 50, p. 4147-4161Research output: Contribution to journal › Journal article › Research › peer-review
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5-substituted imidazole-4-acetic acid analogues: synthesis, modeling, and pharmacological characterization of a series of novel ¿-aminobutyric acidC receptor agonists
Madsen, C., Jensen, A. A., Liljefors, T., Kristiansen, Uffe, Nielsen, Birgitte, Hansen, C. P., Larsen, M., Ebert, B., Bang-Andersen, B., Krogsgaard-Larsen, Povl & Frølund, Bente, 2007, In: Journal of Medicinal Chemistry. 50, 17, p. 4147-4161Research output: Contribution to journal › Journal article › Research › peer-review
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Delineation of the functional properties exhibited by the Zinc-Activated Channel (ZAC) and its high-frequency Thr128Ala variant (rs2257020) in Xenopus oocytes
Madjroh, Nawid, Davies, P. A., Smalley, J. L., Kristiansen, Uffe, Söderhielm, P. C. & Jensen, Anders A., 2021, In: Pharmacological Research. 169, 18 p., 105653.Research output: Contribution to journal › Journal article › Research › peer-review
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Hydroxy-1,2,5-oxadiazolyl moiety as bioisoster of the carboxy function.Synthesis, ionization constants and pharmacological characterization of gamma-aminobutyric acid (GABA) related compounds
Lolli, M. L., Hansen, S. L., Rolando, B., Nielsen, Birgitte, Wellendorph, Petrine, Madsen, K., Larsen, O. M., Kristiansen, Uffe, Fruttero, R., Gasco, A. & Johansen, Tommy Nørskov, 2006, In: J. Med. Chem.. 49, p. 4442-4446 5 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Increasing cellular lifespan with a flow system in organotypic culture of the Laterodorsal Tegmentum (LDT)
Leguizamon, Cesar Ramon Romero, Elnagar, M., Kristiansen, Uffe & Kohlmeier, Kristi Anne, 6 Feb 2019, In: Scientific Reports. p. 1 - 11 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Impaired hippocampal acetylcholine release parallels spatial memory deficits in Tg2576 mice subjected to basal forebrain cholinergic degeneration
Laursen, B., Mørk, A., Plath, N., Kristiansen, Uffe & Bastlund, J. F., 11 Nov 2013, In: Brain Research. 1543, p. 253-262Research output: Contribution to journal › Journal article › Research › peer-review
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Cholinergic degeneration is associated with increased plaque deposition and cognitive impairment in APPswe/PS1dE9 mice
Laursen, B., Mørk, A., Plath, N., Kristiansen, Uffe & Bastlund, J. F., 1 Mar 2013, In: Behavioural Brain Research. 240, 1, p. 146-52 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Hippocampal P3-Like Auditory Event-Related Potentials are Disrupted in a Rat Model of Cholinergic Degeneration in Alzheimer's Disease: Reversal by Donepezil Treatment: Reversal by Donepezil Treatment
Laursen, B., Mørk, A., Kristiansen, Uffe & Bastlund, J. F., 2 Jul 2014, In: Journal of Alzheimer's Disease. 42, 4, p. 1179–1189 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Uterine contraction induced by Ghanaian plants used to induce abortion
Larsen, B. H., Soelberg, Jens, Kristiansen, Uffe & Jäger, A. K., 2016, In: South African Journal of Botany. 106, p. 137-39 3 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Ligands for the GABAA receptor complex
Krogsgaard-Larsen, Povl, Frølund, Bente, Kristiansen, Uffe & Ebert, B., 1 Jan 2001, Glutamate and GABA Receptors and Transporters: Structure, Function and Pharmacology. CRC Press, p. 236-274 39 p.Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
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Novel (Gamma-Aminobutyric Acid)A Agonists and Partial Agonists
Krogsgaard-Larsen, Povl, Frølund, Bente, Kristiansen, Uffe, Lambert, J. D. C., Falch, E. & Curtis, D. R., 1991, Transmitter Amino Acid Receptors. Barnard, E. A. & Costa, E. (eds.). Raven Press, p. 237–249Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
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GABA(A) and GABA(B) receptor agonists, partial agonists, antagonists and modulators: Design and therapeutic prospects
Krogsgaard-Larsen, Povl, Frølund, Bente, Kristiansen, Uffe, Frydenvang, Karla Andrea & Ebert, B., Nov 1997, In: European Journal of Pharmaceutical Sciences. 5, 6, p. 355-384 30 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Ligands for the GABAA receptor complex
Krogsgaard-Larsen, Povl, Frølund, Bente, Kristiansen, Uffe & Ebert, B., 2002, Glutamate and GABA receptors of AMPA/kainate receptors and transporters. Taylor & Francis, p. 236–274Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research
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Ligand Structural Specificity of GABAA Receptors in Guinea Pig Ileum
Kristiansen, Uffe & Fjalland, B., May 1991, In: Pharmacology & Toxicology. 68, 5, p. 332-339 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 985515
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Increasing cellular lifespan with a flow system in organotypic culture of the Laterodorsal Tegmentum (LDT)
Research output: Contribution to journal › Journal article › Research › peer-review
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Discovery of a new class of orthosteric antagonists with nanomolar potency at extrasynaptic GABAA receptors
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Astrocytic GABA transporter activity modulates excitatory neurotransmission
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